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Showing results 1 to 17 of 17

Issue DateTitleAuthor(s)TypeView
2018-10-20A novel TRAP1 inhibitor, containing flexible triphenylphosphonium, interacted with an allosteric site involving E403 residue and triggered protein conformational changesYoon, Nam Gu; Kang, Byoung HeonCONFERENCE190
2020-10-08A novel TRAP1 inhibitor, UB-010 potently inactivates the mitochondrial chaperoneby interacting with the client binding site.Yoon, Nam Gu; Hu, Sung; Kim. So-Yeon; Lee, Changwook; Kang, Byoung HeonCONFERENCE242
2022-02Anticancer strategy targeting the tumor microenvironment and development of potent TRAP1 inhibitorsKang, Byoung Heon; Yoon, Nam GuDoctoral thesis373
2017-04-03Chemical approaches to development of mitochondrial-targeted Hsp90 inhibitor as anti-cancer therapeutics: Mechanism and conformational change of mitochondrial Hsp90Hu, Sung; Yoon, Nam Gu; Kang, Byoung HeonCONFERENCE188
2021-07Design and Synthesis of TRAP1 Selective Inhibitors: H-Bonding with Asn171 Residue in TRAP1 Increases Paralog SelectivityYang, Sujae; Yoon, Nam Gu; Kim, Dongyoung; Park, Eunsun; Kim, So-Yeon; Lee, Ji Hoon; Lee, Changwook; Kang, Byoung Heon; Kang, SoosungARTICLE190
2020-08Development of pyrazolo[3,4-d]pyrimidine-6-amine-based TRAP1 inhibitors that demonstrate in vivo anticancer activity in mouse xenograft modelsKim, Darong; Kim, So-Yeon; Kim, Dongyoung; Yoon, Nam Gu; Yun, Jisu; Hong, Ki Bum; Lee, Changwook; Lee, Ji Hoon; Kang, Byoung Heon; Kang, SoosungARTICLE267
2020-01Discovery of 2-((4-resorcinolyl)-5-aryl-1,2,3-triazol-1-yl)acetates as potent Hsp90 inhibitors with selectivity over TRAP1Jung, Sejin; Yoon, Nam Gu; Yang, Sujae; Kim, Darong; Lee, Won Seok; Hong, Ki Bum; Lee, Changwook; Kang, Byoung Heon; Lee, Ji Hoon; Kang, SoosungARTICLE335
2020-03Dual Binding to Orthosteric and Allosteric Sites Enhances the Anticancer Activity of a TRAP1-Targeting DrugHu, Sung; Ferraro, Mariarosaria; Thomas, Ajesh P.; Chung, Jeong Min; Yoon, Nam Gu; Seol, Ji-Hoon; Kim, Sangpil; Kim, Han-Ul; An, Mi Young; Ok, Haewon; Jung, Hyun Suk; Ryu, Ja-Hyoung; Colombo, Giorgio; Kang, Byoung HeonARTICLE350
2020-10-08Function of mitochondrial HSP90 in tumor angiogenesisKim, So Yeon; Yoon, Nam Gu; Kim, Eun Hye; Kang, Byoung HeonCONFERENCE226
2021-12-10Function of mitochondrial HSP90 in tumor microenvironmentKim, So Yeon; Yoon, Nam Gu; Kang, Byoung HeonCONFERENCE373
2021-08-25Function of mitochondrial HSP90 in tumor micronenvironmentKim, So Yeon; Yoon, Nam Gu; Kang, Byoung HeonCONFERENCE84
2021-12-10MitoQ inactivates mitochondrial chaperone TRAP1 by interacting with the client binding siteYoon, Nam Gu; Kang, Byoung HeonCONFERENCE376
2021-12Mitoquinone Inactivates Mitochondrial Chaperone TRAP1 by Blocking the Client Binding SiteYoon, Nam Gu; Lee, Hakbong; Kim, So-Yeon; Hu, Sung; Kim, Darong; Yang, Sujae; Hong, Ki Bum; Lee, Ji Hoon; Kang, Soosung; Kim, Byung-Gyu; Myung, Kyungjae; Lee, Changwook; Kang, Byoung HeonARTICLE243
2022-03Quaternary ammonium-based mitochondria targeting anticancer agents with high water solubilityKim, Sangpil; Yoon, Nam Gu; Jana, Batakrishna; Kang, Byoung Heon; Ryu, Ja-HyoungARTICLE58
2021-08-25SMx inactivates mitochondrial chaperone TRAP1 by interacting with the client binding siteYoon, Nam Gu; Kang, Byoung HeonCONFERENCE64
2022-09Triphenylphosphonium conjugation to a TRAP1 inhibitor, 2-amino-6--chloro-7,9-dihydro-8H-purin-8-one increases antiproliferative activityYang, Sujae; Yoon, Nam Gu; Park, Min-A; Yun, Jisu; Im, Jin Young; Kang, Byoung Heon; Kang, SoosungARTICLE178
2020-01Unleashing the full potential of Hsp90 inhibitors as cancer therapeutics through simultaneous inactivation of Hsp90, Grp94, and TRAP1Park, Hye-Kyung; Yoon, Nam Gu; Lee, Ji-Eun; Hu, Sung; Yoon, Sora; Kim, So Yeon; Hong, Jun-Hee; Nam, Dougu; Chae, Young Chan; Park, Jong Bae; Kang, Byoung HeonARTICLE501
Showing results 1 to 17 of 17

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